产品编号:X750948
产品规格:2.5mg
产品价格:面议
| 标准品编号: | X750948 |
| 名称: | XMD 8-92 |
| 别名: | 2-[[2-Ethoxy-4-(4-hydroxy-1-piperidinyl)phenyl]amino]-5,11-dihydro-5,11-dimethyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one |
| CAS号: | 1234480-50-2 |
| 分子式: | C₂₆H₃₀N₆O₃ |
| 分子量: | 474.55 |
| 类别: | Standards; Pharmaceutical/API Drug Impurities/Metabolites; |
| 应用: | XMD 8-92, is a BMK1 inhibitor and a highly selective inhibitor of ERK5 activity. XMD8-92 blocks cellular BMK1 activation and significantly suppresses tumor growth in lung and cervical tumor models and is well tolerated in animals. |
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