XMD 8-92

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产品编号:X750948

产品规格:2.5mg

产品价格:面议


产品详情

标准品编号: X750948
名称: XMD 8-92
别名: 2-[[2-Ethoxy-4-(4-hydroxy-1-piperidinyl)phenyl]amino]-5,11-dihydro-5,11-dimethyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
CAS号: 1234480-50-2
分子式: C₂₆H₃₀N₆O₃
分子量: 474.55
类别: Standards; Pharmaceutical/API Drug Impurities/Metabolites;
应用: XMD 8-92, is a BMK1 inhibitor and a highly selective inhibitor of ERK5 activity. XMD8-92 blocks cellular BMK1 activation and significantly suppresses tumor growth in lung and cervical tumor models and is well tolerated in animals.
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