E 7449

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产品编号:E102500

产品规格:5mg

产品价格:面议


产品详情

标准品编号: E102500
名称: E 7449
别名: 8-[(1,3-Dihydro-2H-isoindol-2-yl)methyl]-1,2-dihydro-3H-pyridazino[3,4,5-de]quinazolin-3-one;
CAS号: 1140964-99-3
分子式: C₁₈H₁₅N₅O
分子量: 317.34
种类: Standards; Enzyme Activators and Inhibitors;
应用: E 7449 is a dual inhibitor of PARP1/2 and tankyrase1/2 exhibits anti-tumor activity in BRCVIP(LA)deficient in vivo models. PARP1/2 and tankyrase1/2 are involved with DNA damage and canonical Wnt/β-catenin signaling, respectively.
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