产品编号:A627960
产品规格:50mg
产品价格:面议
| 标准品编号: | A627960 |
| 名称: | Trelagliptin Trifluoroacetic Acid Salt |
| 别名: | 2-[[6-[(3R)-3-Amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-4-fluorobenzonitrile Trifluoroacetic Acid Salt |
| CAS号: | 928201-45-0 |
| 备用CAS: | 865759-25-7-for free base |
| 分子式: | C₂₀H₂₁F₄N₅O₄ |
| 分子量: | 471.41 |
| 类别: | Standards; Pharmaceutical/API Drug Impurities/Metabolites; |
| 应用: | 2-[[6-[(3R)-3-Amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-4-fluorobenzonitrile trifluoroacetic acid salt is a potent, selective, and noncovalent inhibitor of dipeptidyl peptidase IV (DPP-4). This inhibitor provides sustained reduction of plasma DPP-4 activity and lowering of blood glucose in animal models of diabetes. |
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