产品名称:Everolimus, Cyclosporine and Tacrolimus Mix Standard
产品CAS:
规格含量:25mg
产品价格:面议
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产品详细介绍
标准品编号:
E608165
名称:
Everolimus, Cyclosporine and Tacrolimus Mix Standard
分子式:
C₅₃H₈₃NO₁₄ • C₆₂H₁₁₁N₁₁O₁₂ • C₄₄H₆₉N
分子量:
958.2212026
种类:
Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
应用:
Everolimus (E945400) is a derivative of Rapamycin. Everolimus inhibits cytokine-mediated lymphocyte proliferation. Cyclosporine(C990065) is an immunopsupressent thought to bind to cyclophilin in T-lymphocytes. Tacrolimus (F370000) is also an immunosuppressant that blocks T-cell proliferation in vitro by inhibiting the generation of several lymphokines, especially IL-2. Shown to inhibit the activity of FK-506 binding protein, thereby reversing its effects on sarcoplasmic reticulum Ca+2 release.