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产品基本信息
产品编号：G797515
产品名称：GSK2656157
产品CAS：1337532-29-2
规格含量：50mg
产品价格：面议
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产品详细介绍
标准品编号:
G797515
名称:
GSK2656157
别名:
1-[5-(4-Amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydro-1H-indol-1-yl]-2-(6-methyl-2-pyridinyl)-ethanone; 5-[4-Fluoro-1-[(6-methyl-2-pyridinyl)acetyl]-2,3-dihydro-1H-indol-5-yl]-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS号:
1337532-29-2
分子式:
C₂₃H₂₁FN₆O
外观:
白色至淡黄色固体
熔点:
194-196°C
分子量:
416.45
储存:
-20°C Freezer
溶解度:
DMSO (Slightly), Methanol (Slightly)
种类:
Standards; Enzyme Activators and Inhibitors;
应用:
GSK2656157 is an ATP-competitive and highly selective inhibitor of PKR-like endoplasmic reticulum kinase (PERK) enzyme activity. GSK2656157 also has anti-tumor and anti-angiogenic activity.
参考文献
Axten, J.M., et al.: ACS Med. Chem. Lett., 4, 964 (2013); Atkins, C., et al.: Cancer Res., 73, 1993 (2013)
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