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Linsitinib-d3
产品基本信息
产品编号:L469022
产品名称:Linsitinib-d3
产品CAS:
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产品价格:面议
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产品详细介绍
标准品编号: L469022
名称: Linsitinib-d3
别名: cis-3-[8-Amino-1-(2-phenyl-7-quinolinyl)imidazo[1,5-a]pyrazin-3-yl]-1-(methyl-d3)cyclobutanol; OSI 906-d3; OSI 906AVIP(LA)d3;
参考CAS号: 类似: 867160-71-2
分子式: C₂₆H₂₀D₃N₅O
分子量: 424.51
种类: Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
应用: Labelled Linsitinib (L469020). Linsitinib is a small-molecule dual insulin-like growth factor-1 receptor (IGF-IR) and insulin receptor (IR) kinase inhibitor. IGF-I receptor (IGF-IR) has been implicated in the promotion of tumorigenesis, metastasis and resistance to cancer therapies and thus Linsitinib may be a useful anticancer agent.
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